Wani, Imtiyaz Ahmad ; Goswami, Gaurav ; Sk, Sahid ; Mal, Abhijit ; Sayyad, Masthanvali ; Ghorai, Manas K. (2020) A synthetic route to 1,4-disubstituted tetrahydro-β-carbolines and tetrahydropyranoindoles via ring-opening/Pictet–Spengler reaction of aziridines and epoxides with indoles/aldehydes Organic & Biomolecular Chemistry, 18 (2). pp. 272-287. ISSN 1477-0520
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Official URL: http://doi.org/10.1039/C9OB02098E
Related URL: http://dx.doi.org/10.1039/C9OB02098E
Abstract
A simple and efficient synthetic route to various 1,4-disubstituted tetrahydro-β-carbolines and tetrahydropyrano[3,4-b]indoles in high yields and stereoselectivity via LiClO4-catalyzed SN2-type ring opening of aziridines and epoxides with indoles followed by p-toluenesulfonic acid (PTSA) catalyzed Pictet–Spengler reaction is described.
| Item Type: | Article |
|---|---|
| Source: | Copyright of this article belongs to Royal Society of Chemistry. |
| ID Code: | 117079 |
| Deposited On: | 15 Apr 2021 07:40 |
| Last Modified: | 15 Apr 2021 07:40 |
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