Items where Author is "Sriram, Dharmarajan"

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Number of items: 23.

Article

Dhameliya, Tejas M. ; Patel, Kshitij I. ; Tiwari, Rishu ; Vagolu, Siva Krishna ; Panda, Dulal ; Sriram, Dharmarajan ; Chakraborti, Asit K. (2021) Design, synthesis, and biological evaluation of benzo[d]imidazole-2-carboxamides as new anti-TB agents Bioorganic Chemistry, 107 . p. 104538. ISSN 00452068

Jadhavar, Pradeep S. ; Patel, Kshitij I. ; Dhameliya, Tejas M. ; Saha, Nirjhar ; Vaja, Maulikkumar D. ; Krishna, Vagolu Siva ; Sriram, Dharmarajan ; Chakraborti, Asit K. (2020) Benzimidazoquinazolines as new potent anti-TB chemotypes: Design, synthesis, and biological evaluation Bioorganic Chemistry, 99 . p. 103774. ISSN 00452068

Bhagat, Srikant ; Supriya, Metheku ; Pathak, Satish ; Sriram, Dharmarajan ; Chakraborti, Asit K. (2019) α-Sulfonamidophosphonates as new anti-mycobacterial chemotypes: Design, development of synthetic methodology, and biological evaluation Bioorganic Chemistry, 82 . pp. 246-252. ISSN 00452068

Dhameliya, Tejas M. ; Tiwari, Rishu ; Banerjee, Arkaprabha ; Pancholia, Sahaj ; Sriram, Dharmarajan ; Panda, Dulal ; Chakraborti, Asit K. (2018) Benzo[d]thiazole-2-carbanilides as new anti-TB chemotypes: Design, synthesis, biological evaluation, and structure-activity relationship European Journal of Medicinal Chemistry, 155 . pp. 364-380. ISSN 02235234

Beesetti, Hemalatha ; Tyagi, Poornima ; Medapi, Brahmam ; Krishna, Vagolu Siva ; Sriram, Dharmarajan ; Khanna, Navin ; Swaminathan, Sathyamangalam (2018) A quinoline compound inhibits the replication of dengue virus serotypes 1–4 in Vero cells Antiviral Therapy, 23 (5). pp. 385-394. ISSN 1359-6535

Pancholia, Sahaj ; Dhameliya, Tejas M. ; Shah, Parth ; Jadhavar, Pradeep S. ; Sridevi, Jonnalagadda Padma ; Yogeshwari, Perumal ; Sriram, Dharmarajan ; Chakraborti, Asit K. (2016) Benzo[d]thiazol-2-yl(piperazin-1-yl)methanones as new anti-mycobacterial chemotypes: design, synthesis, biological evaluation and 3D-QSAR studies European Journal of Medicinal Chemistry, 116 . pp. 187-199. ISSN 0223-5234

Jadhavar, Pradeep S. ; Dhameliya, Tejas M. ; Vaja, Maulikkumar D. ; Kumar, Dinesh ; Sridevi, Jonnalagadda Padma ; Yogeeswari, Perumal ; Sriram, Dharmarajan ; Chakraborti, Asit K. (2016) Synthesis, biological evaluation and structure–activity relationship of 2-styrylquinazolones as anti-tubercular agents Bioorganic & Medicinal Chemistry Letters, 26 (11). pp. 2663-2669. ISSN 0960-894X

Suryadevara, Priyanka ; Perumal, Yogeeswari ; Soni, Vijay ; Parthiban, Brindha Devi ; Nandicoori, Vinay Kumar ; Sriram, Dharmarajan (2016) Computational sampling and simulation based assessment of novel Mycobacterium tuberculosis glutamine synthetase inhibitors: Study involving structure based drug design and free energy perturbation Current Topics in Medicinal Chemistry, 16 (9). pp. 978-995. ISSN 1568-0266

Tanwar, Babita ; Kumar, Asim ; Yogeeswari, Perumal ; Sriram, Dharmarajan ; Chakraborti, Asit K. (2016) Design, development of new synthetic methodology, and biological evaluation of substituted quinolines as new anti-tubercular leads Bioorganic & Medicinal Chemistry Letters, 26 (24). pp. 5960-5966. ISSN 0960894X

Banerjee, Srijon Kaushik ; Kumar, Manish ; Alokam, Reshma ; Sharma, Arun Kumar ; Chatterjee, Ayan ; Kumar, Ranjeet ; Sahu, Sanjaya Kumar ; Jana, Kuladip ; Singh, Ramandeep ; Yogeeswari, Perumal ; Sriram, Dharmarajan ; Basu, Joyoti ; Kundu, Manikuntala (2016) Targeting multiple response regulators of Mycobacterium tuberculosis augments the host immune response to infection Scientific Reports, 6 (1). ISSN 2045-2322

Soni, Vijay ; Suryadevara, Priyanka ; Sriram, Dharmarajan ; Kumar, Santhosh ; Nandicoori, Vinay Kumar ; Yogeeswari, Perumal (2015) Structure-based design of diverse inhibitors of Mycobacterium tuberculosis N-acetylglucosamine-1-phosphate uridyltransferase: combined molecular docking, dynamic simulation and biological activity Journal of Molecular Modeling, 21 (7). 1Article ID 74. ISSN 1610-2940

Soni, Vijay ; Upadhayay, Sandeep ; Suryadevara, Priyanka ; Samla, Ganesh ; Singh, Archana ; Yogeeswari, Perumal ; Sriram, Dharmarajan ; Nandicoori, Vinay Kumar (2015) Depletion of M. tuberculosis GlmU from infected murine lungs effects the clearance of the pathogen PLoS Pathogens, 11 (10). pp. Article ID e1005235-27 pages. ISSN 1553-7366

Shah, Parth ; Dhameliya, Tejas M. ; Bansal, Rohit ; Nautiyal, Manesh ; Kommi, Damodara N. ; Jadhavar, Pradeep S. ; Sridevi, Jonnalagadda Padma ; Yogeeswari, Perumal ; Sriram, Dharmarajan ; Chakraborti, Asit K. (2014) N-arylalkylbenzo[d]thiazole-2-carboxamides as anti-mycobacterial agents: design, new methods of synthesis and biological evaluation MedChemComm, 5 (10). pp. 1489-1495. ISSN 2040-2503

Senthilkumar, Palaniappan ; Dinakaran, Murugesan ; Yogeeswari, Perumal ; China, Arnab ; Nagaraja, V. ; Sriram, Dharmarajan (2009) Antimycobacterial activities of novel fluoroquinolones Biomedicine & Pharmacotherapy, 63 (1). pp. 27-35. ISSN 0753-3322

Senthilkumar, Palaniappan ; Dinakaran, Murugesan ; Yogeeswari, Perumal ; Sriram, Dharmarajan ; China, Arnab ; Nagaraja, Valakunja (2009) Synthesis and antimycobacterial activities of novel 6-nitroquinolone-3-carboxylic acids European Journal of Medicinal Chemistry, 44 (1). pp. 345-358. ISSN 0223-5234

Dinakaran, Murugesan ; Senthilkumar, Palaniappan ; Yogeeswari, Perumal ; China, Arnab ; Nagaraja, Valakunja ; Sriram, Dharmarajan (2008) Synthesis, antimycobacterial activities and phototoxic evaluation of 5H-thiazolo[3,2-a]quinoline-4-carboxylic acid derivatives Medicinal Chemistry, 4 (5). pp. 482-491. ISSN 1573-4064

Murugesan, Dinakaran ; Palaniappan, Senthilkumar ; Perumal, Yogeeswari ; Arnab, China ; Valakunja, Nagaraja ; Sriram, Dharmarajan (2008) Antimycobacterial and phototoxic evaluation of novel 6-fluoro/nitro-4-oxo-7-(sub)-4H-[1,3]thiazeto[3,2-a]quinoline-3-carboxylic acid International Journal of Antimicrobial Agents, 31 (4). pp. 337-344. ISSN 0924-8579

Dinakaran, Murugesan ; Senthilkumar, Palaniappan ; Yogeeswari, Perumal ; China, Arnab ; Nagaraja, Valakunja ; Sriram, Dharmarajan (2008) Antimycobacterial activities of novel 2-(sub)-3-fluoro/nitro-5,12-dihydro-5-oxobenzothiazolo[3,2-a]quinoline-6-carboxylic acid Bioorganic & Medicinal Chemistry, 16 (6). pp. 3408-3418. ISSN 0968-0896

Senthilkumar, Palaniappan ; Dinakaran, Murugesan ; Banerjee, Debjani ; Devakaram, Ruth Vandana ; Yogeeswari, Perumal ; China, Arnab ; Nagaraja, Valakunja ; Sriram, Dharmarajan (2008) Synthesis and antimycobacterial evaluation of newer 1-cyclopropyl-1,4-dihydro-6-fluoro-7-(substituted secondary amino)-8-methoxy-5-(sub)-4-oxoquinoline-3-carboxylic acids Bioorganic & Medicinal Chemistry, 16 (5). pp. 2558-2569. ISSN 0968-0896

Dinakaran, Murugesan ; Senthilkumar, Palaniappan ; Yogeeswari, Perumal ; China, Arnab ; Nagaraja, Valakunja ; Sriram, Dharmarajan (2008) Novel ofloxacin derivatives: synthesis, antimycobacterial and toxicological evaluation Bioorganic & Medicinal Chemistry Letters, 18 (3). pp. 1229-1236. ISSN 0960-894X

Sriram, Dharmarajan ; Senthilkumar, Palaniappan ; Dinakaran, Murugesan ; Yogeeswari, Perumal ; China, Arnab ; Nagaraja, Valakunja (2007) Antimycobacterial activities of novel 1-(cyclopropyl/tert-butyl/4-fluorophenyl)-1,4-dihydro- 6-nitro-4-oxo-7-(substituted secondary amino)-1,8-naphthyridine-3-carboxylic acid Journal of Medicinal Chemistry, 50 (24). pp. 6232-6239. ISSN 0022-2623

Sriram, Dharmarajan ; Bal, Tanushree Ratan ; Yogeeswari, Perumal ; Radha, Deshpande R. ; Nagaraja, Valakunja (2006) Evaluation of antimycobacterial and DNA gyrase inhibition of fluoroquinolone derivatives Journal of General and Applied Microbiology, 52 (4). pp. 195-200. ISSN 0022-1260

Sriram, Dharmarajan ; Yogeeswari, Perumal ; Basha, Jafar Sadik ; Radha, Deshpande R. ; Nagaraja, Valakunja (2005) Synthesis and antimycobacterial evaluation of various 7-substituted ciprofloxacin derivatives Bioorganic & Medicinal Chemistry, 13 (20). pp. 5774-5778. ISSN 0968-0896

This list was generated on Sat Apr 4 09:18:37 2026 UTC.