Items where Author is "De Lombaert, Stephane"

Article

Blum, Charles A. ; Zheng, Xiaozhang ; Brielmann, Harry ; Hodgetts, Kevin J. ; Bakthavatchalam, Rajagopal ; Chandrasekhar, Jayaraman ; Krause, James E. ; Cortright, Daniel ; Matson, David ; Crandall, Marci ; Ngo, Chu K. ; Fung, Lawrence ; Day, Marta ; Kershaw, Mark ; De Lombaert, Stephane ; Chenard, Bertrand L. (2008) Aminoquinazolines as TRPV1 antagonists: modulation of drug-like properties through the exploration of 2-position substitution Bioorganic & Medicinal Chemistry Letters, 18 (16). pp. 4573-4577. ISSN 0960-894X

Yoon, Taeyoung ; De Lombaert, Stephane ; Brodbeck, Robbin ; Gulianello, Michael ; Chandrasekhar, Jayaraman ; Horvath, Raymond F. ; Ge, Ping ; Kershaw, Mark T. ; Krause, James E. ; Kehne, John ; Hoffman, Diane ; Doller, Dario ; Hodgetts, Kevin J. (2008) The design, synthesis and structure-activity relationships of 1-aryl-4-aminoalkylisoquinolines: a novel series of CRF-1 receptor antagonists Bioorganic & Medicinal Chemistry Letters, 18 (3). pp. 891-896. ISSN 0960-894X

Zheng, Xiaozhang ; Hodgetts, Kevin J. ; Brielmann, Harry ; Hutchison, Alan ; Burkamp, Frank ; Jones, A. Brian ; Blurton, Peter ; Clarkson, Robert ; Chandrasekhar, Jayaraman ; Bakthavatchalam, Rajagopal ; De Lombaert, Stephane ; Crandall, Marci ; Cortright, Daniel ; Blum, Charles A. (2006) From arylureas to biarylamides to aminoquinazolines: discovery of a novel, potent TRPV1 antagonist Bioorganic & Medicinal Chemistry Letters, 16 (19). pp. 5217-5221. ISSN 0960-894X